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Histone Acetyltransferase Inhibitor II
Histone Acetyltransferase Inhibitor II
CAS No. 932749-62-7
Histone Acetyltransferase Inhibitor II ( —— )
Catalog No. M22025 CAS No. 932749-62-7
Histone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
5MG | 65 | In Stock |
|
10MG | 99 | In Stock |
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25MG | 195 | In Stock |
|
50MG | 336 | In Stock |
|
100MG | 500 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
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Product NameHistone Acetyltransferase Inhibitor II
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NoteResearch use only, not for human use.
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Brief DescriptionHistone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells.
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DescriptionHistone Acetyltransferase Inhibitor II is a selective and cell permeable inhibitor of p300 histone acetyltransferase(IC50 : 5 μM).with anti-acetylase activity in mammalian cells. Histone Acetyltransferase Inhibitor II (compound 2c) was the most active inhibitor, also showing high specificity for p300 as compared to other histone acetyltransferases.?Most notably, 2c showed anti-acetylase activity in mammalian cells.
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetEpigenetic Reader Domain
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Recptorp300
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Research Area——
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Indication——
Chemical Information
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CAS Number932749-62-7
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Formula Weight464.15
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Molecular FormulaC20H16Br2O3
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Purity>98% (HPLC)
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SolubilityDMSO:30 mg/mL (64.63 mM)
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SMILESC1CC(=CC2=CC(=C(C=C2)O)Br)C(=O)C(=CC3=CC(=C(C=C3)O)Br)C1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Costi R, et al. Cinnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase. J Med Chem. 2007 Apr 19;50(8):1973-7. Epub 2007 Mar 10.
molnova catalog
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